Статьи 2004

Frolov, E. B.; Lakner, F. J.; Khvat, A. V.; Ivachtchenko, A. V. An efficient synthesis of novel 1,3-oxazolo[4,5-d]pyridazinones. Tetrah. Lett., 45(24), 4693–4696 (2004). 

Okun, I.; Balakin, K. V.; Savchuk, N. P. Focused versus random screening for abl kinase inhibitors. Current Drug Disc. 9, 15-18 (2004). 

Savchuk, N. P.; Balakin, K. V. An efficient primary hit optimization strategy. Current Drug Disc. 5, 23-27 (2004). 

Savchuk, N. P.; Balakin, K. V.; Tkachenko, S. E. Exploring the chemogenomic knowledge space with annotated chemical libraries. Curr. Opin. Chem. Biol., 8(4), 412–417 (2004). 

Ivachtchenko, A. V.; Khvat, A. V.; Kobak, V. V.; Kysil, V. M.; Williams, C. T. A new insight into the Pfitzinger reaction. A facile synthesis of 6-sulfamoylquinoline-4-carboxylic acids. Tetrah. Lett., 45(28), 5473–5476 (2004). 

Ivachtchenko, A. V.; Khvat, A. V.; Tkachenko, S. E.; Sandulenko, Yu. B.; Vvedensky, V. Y. Access to novel substituted diazaadamantanes via semi-natural tetrahydrocytisine. Tetrah. Lett., 45(36), 6733–6736 (2004). 

Ivachtchenko, A.; Kovalenko, S.; Tkachenko, O. V.; Parkhomenko, O. Synthesis of Substituted Thienopyrimidine-4-ones. J. Combin. Chem., 6(4), 573–583 (2004). 

Ivachtchenko, A. V.; Tkachenko, S. E.; Sandulenko, Yu. B.; Vvedensky, V. Y. Khvat, A. V.; A Parallel Solution-Phase Synthesis of Substituted 3,7-Diazabicyclo[3.3.1]nonanes. J. Combin. Chem., 6(5), 828–834 (2004). 

Zhuravel, I. O.; Kovalenko, S. M.; Ivachtchenko, A. V.; Chernykh, V. P.; Shinkarenko, P. E. Synthesis of substituted 3-(5-amino-[1,3,4]thiadiazol-2-yl)-2H-pyrano[2,3-c]pyridin-2-ones. J. Heterocycl. Chem., 41(4), 517–524 (2004). 

Ivachtchenko, A. V.; Kravchenko, D. V.; Zheludeva, V. I.; Pershin, D. G. Synthesis of pinacol esters of 1-alkyl-1H-pyrazol-5-yl- and 1-alkyl-1H-pyrazol-4-ylboronic acids. J. Heterocycl. Chem., 41(6), 931–939 (2004). 

Dorogov, M. V.; Filimonov, S. I.; Kobylinsky, D. B.; Ivanovsky S. A.; Korikov, P. V.; Soloviev, M. Y.; Khahina, M. Y.; Shalygina, E. E.; Kravchenko, D. V.; Ivachtchenko, A. V. A convenient synthesis of novel 3-(heterocyclylsulfonyl)propanoic acids and their amide derivatives. Synthesis, 2999–3004 (2004). 

Silin, O. V.; Savchenko, T. I.; Kovalenko, S, M.; Nikitchenko, V. M.; Ivachtchenko, A. V. Synthesis of 5H-pyrazolo[4,3-c]quinolines. Heterocycles, 63(8), 1883–1890 (2004). 

Заложнев, А. Ю.; Иващенко, А. А.; Овчинникова Т. И. Модели и методы управления развитием фирмы. Сист. управ. информ. технол., 38–41 (2004). 

Иващенко, А. А.; Матвеев, А. А.; Новиков, Д. А.; Сухачев, К. А. Институциональное и мотивационное управление организационными системами. Сборник трудов IV Международной конференции «Современные сложные системы управления». Тверь, ТГТУ, 299–302 (2004). 

Tkachenko, S. E.; Okun, I.; Balakin, K. V.; Petersen, C. E.; Ivanenkov, Y. A.; Savchuk, N. P.; Ivashchenko, A. A. Efficient optimization strategy for marginal hits active against abl tyrosine kinases. Curr. Drug Discov. Techn., 1(3), 201–210 (2004). 

Balakin, K. V.; Ekins, S.; Bugrim, A.; Ivanenkov, Y. A.; Korolev, D.; Nikolsky, Y. V.; Ivashchenko, A. A.; Savchuk, N. P.; Nikolskaya, T. Quantitative structure-metabolism relationship modeling of metabolic N-dealkylation reaction rates. Drug Metabol. Disp., 32(10), 1111–1120 (2004). 

Balakin, K. V.; Ekins, S.; Bugrim, A.; Ivanenkov, Y. A.; Korolev, D.; Nikolsky, Y. V.; Skorenko, A. V.; Ivashchenko, A. A.; Savchuk, N. P.; Nikolskaya, T. Kohonen maps for prediction of binding to human cytochrome P450 3A4. Drug Metabol. Disp., 32(10), 1183–1189 (2004). 

Balakin, K. V.; Tkachenko, S. E.; Okun, I.; Skorenko, A. V.; Ivanenkov, Y. A.; Savchuk, N. P.; Ivashchenko, A. A.; Nikolsky, Y. Bioisosteric morphing in primary hit optimization. Chim. Oggi, 22(1–2), 15–18 (2004). 

Balakin, K. V.; Ivanenkov, Y. A.; Skorenko, A. V.; Nikolsky, Y. V.; Savchuk, N.P.; Ivashchenko, A. A. In silico estimation of DMSO solubility of organic compounds for bioscreening. J. Biomol. Scr., 9(1), 22–31 (2004).